The role of PDE-4 in neurodegenerative disorders

  • Research type

    Research Study

  • Full title

    The role of PDE-4 in neurodegenerative disorders: An 11C-rolipram PET study in Parkinson’s and Huntington’s disease

  • IRAS ID

    162128

  • Contact name

    Marios Politis

  • Contact email

    marios.politis@kcl.ac.uk

  • Sponsor organisation

    King's College London

  • Duration of Study in the UK

    3 years, 0 months, 1 days

  • Research summary

    Phosphodiesterase 4 (PDE-4) is a protein expressed in a specific area of the brain called striatum, which contribute to the control of movement and behaviour. Previous work on animals have shown that dysregulation of PDE-4 may lead cells in the brain to die. Parkinson’s (PD) and Huntington’s (HD) disease are two progressive neurological conditions, which affect mainly the striatum. PDE-4 could be a key therapeutic target in HD and PD, however its expression and importance in humans is unknown. Previous animal studies have shown that PDE-4 inhibition with rolipram can lead to a decrease of neuronal loss in the striatum of animal model of HD. In this study, we aim to investigate in vivo the expression of PDE-4 enzyme in PD patients and HD gene carriers using positron emission tomography (PET) with 11C-rolipram, which is a specific tracer for PDE-4. We hypothesise that PDE-4 will be dysregulated in specific areas of the brain relevant to the control of movements playing a critical role in neurodegeneration.

  • REC name

    London - Bromley Research Ethics Committee

  • REC reference

    14/LO/2104

  • Date of REC Opinion

    26 Nov 2014

  • REC opinion

    Favourable Opinion