PLN-74809: Safety, tolerability and cardiodynamics of SAD

  • Research type

    Research Study

  • Full title

    A Continued Evaluation of the Safety, Tolerability, and Cardiodynamics of Single Ascending Doses of PLN-74809 in Healthy Participants.

  • IRAS ID

    1006689

  • Contact name

    Annie Clark

  • Contact email

    aclark@pliantrx.com

  • Sponsor organisation

    Pliant Therapeutics Inc

  • ISRCTN Number

    ISRCTN67246142

  • Research summary

    A double blind study to assess the safety, tolerability, and effect of the heart of a single ascending dose of the IMP (PLN-74809).The clinical trial investigational medicine, PLN-74809 is experimental. That means the Medicines and Health Care Regulatory Agency (MHRA) has not approved it for use outside the clinical trials. PLN-74809 is being studied to treat Idiopathic Pulmonary Fibrosis which is a condition in which tiny air sacs in the lungs become damaged, causing build-up of scar tissue and Primary Sclerosing Cholangitis which is a rare disease that attacks the bile ducts causing your liver bile ducts to become scarred. \nThe entire clinical trial duration is about 15 days plus up to 28 days for screening (running investigations on bloods, vital signs, ECG, etc.. to confirm eligibility of the participant to enrol into the study). There is a confinement period of about 8 days. There is 1 outpatient return visit to the clinic.\nEach volunteer will be enrolled into a specific dose level group. In each group, participants will be randomly assigned (by chance like flipping a coin) to receive PLN-74809 or placebo. Out of 60 subjects, 40 will receive PLN-74809 and 20 will receive placebo. A placebo is a tablet that looks like PLN-7408 but contains no investigational medicine. The use of a placebo helps to make sure that any side effects during the clinical trial are judged fairly. \nDose Level 1: 960 mg single dose of PLN-74809 or placebo\nDose Level 2: 1360 mg single dose of PLN-74809 or placebo\nDose Level 3: 1920 mg single dose of PLN-74809 or placebo\nDose Level 4: 2640 mg single dose of PLN-74809 or placebo\t\nDose Level 5: To be determined \nThe Clinical trial Doctor and the Sponsor will review the safety data of each dose level. The next dose level will not be dosed until the safety data has been reviewed. The Sponsor and/or the Clinical trial Doctor can stop the clinical trial at any time.

  • REC name

    London - London Bridge Research Ethics Committee

  • REC reference

    22/LO/0842

  • Date of REC Opinion

    21 Mar 2023

  • REC opinion

    Further Information Favourable Opinion