PK of Modified Release formulations of GSK2982772 (QCL117918)

  • Research type

    Research Study

  • Full title

    A two part, non-randomised, open label study designed to assess the pharmacokinetics of GSK2982772 following administration of modified release formulations in capsule relative to an immediate release reference tablet formulation (Part A) and the pharmacokinetics of escalating, repeat doses of a selected modified release prototype (Part B) in healthy subjects

  • IRAS ID

    229633

  • Contact name

    Dipak Kothari

  • Contact email

    dipak.p.kothari@gsk.com

  • Sponsor organisation

    GlaxoSmithKline Research & Development Limited

  • Eudract number

    2017-000652-25

  • Duration of Study in the UK

    0 years, 4 months, 13 days

  • Research summary

    The sponsor GlaxoSmithKline Research & Development Limited (also known as GSK) are developing a new formulation (recipe) of the test medicine GSK2982772, for the potential treatment of diseases caused by inflammation such as inflammatory bowel disease (IBD), plaque psoriasis (PsO), rheumatoid arthritis (RA).

    The study will try to identify a new formulation of the test medicine which allows for more convenient once daily dosing for patients.

    The study will consist of 2 parts. Part A is a 6 period cross-over in 16 healthy volunteers, designed to evaluate up to 4 formulations following single 120 mg doses in the fasted state. This part may also investigate the effect of food on a selected formulation, and there is also the option to cancel Periods 5 and 6 if favourable formulation is determined in Periods 1 or 2. Part B is a 3 period cross-over in 10 healthy volunteers designed to evaluate 3 days of repeat dosing of a selected formulation of the test medicine at target daily doses of 30, 60 and 240 mg given either once or twice day.

  • REC name

    South Central - Berkshire B Research Ethics Committee

  • REC reference

    17/SC/0404

  • Date of REC Opinion

    5 Sep 2017

  • REC opinion

    Further Information Favourable Opinion