*Open-Label PET Study Investigating ENX-104

  • Research type

    Research Study

  • Full title

    An open-label positron emission tomography (PET) study to demonstrate safety, tolerability, receptor occupancy, and pharmacokinetics after a single oral dose administration of ENX-104 in healthy volunteers

  • IRAS ID

    1010977

  • Contact name

    Eve Taylor

  • Contact email

    eve.taylor@engrail.com

  • Sponsor organisation

    Engrail Therapeutics, Inc.

  • Clinicaltrials.gov Identifier

    NCT07253272

  • Research summary

    The trial is a single centre, open-label trial in up to 10 healthy, non-smoking males and females assigned at birth, inclusive of any gender identity between the ages of 23 and 65 years. \n\nThe medicine to be tested is this trial is a compound called ENX-104 being developed a new therapy for treating major depressive disorder and/or other disorders of the central nervous system (CNS).\n\nThe main purpose of the clinical trial is to see how safe the clinical trial medicine is and how well it is tolerated after dosing of the clinical trial medicine in healthy subjects and how it is absorbed in the brain. The clinical trial will also investigate how the clinical trial medicine is taken up and metabolised (chemically broken down). \nThe trial will comprise of:\n-\tScreening period of a maximum 45 days – Day -45 to Day -1\n-\tIn-house Treatment Period - Day -2 to Day 2 (admission on Day -2, Dosing on Day 1)\n-\tA Follow up Visit on Day 9

  • REC name

    London - Brent Research Ethics Committee

  • REC reference

    24/LO/0813

  • Date of REC Opinion

    13 Jan 2025

  • REC opinion

    Further Information Favourable Opinion