Investigate Safety, Tolerability & Pharmacokinetics of Inhaled AZD0449

  • Research type

    Research Study

  • Full title

    A Single blind, Randomized, Placebo-controlled Three part Study in Healthy Volunteers and Patients with Mild Asthma to Investigate the Safety, Tolerability and Pharmacokinetics of Inhaled AZD0449 Following Single and Multiple Ascending Doses and to Investigate the Anti-inflammatory Effect of Inhaled AZD0449

  • IRAS ID

    250847

  • Contact name

    Pablo ForteSoto

  • Contact email

    Pablo.ForteSoto@parexel.com

  • Sponsor organisation

    AstraZeneca

  • Eudract number

    2018-003469-32

  • Duration of Study in the UK

    1 years, 1 months, 18 days

  • Research summary

    Summary of Research
    This is a single-blind, randomised, placebo-controlled, three-part study to investigate the safety, tolerability, pharmacokinetics (PK) and the anti-inflammatory effect of AZD0449 in healthy volunteers (Part 1) and patients with mild asthma (Parts 2 and 3). AZD0449 is a potentially new asthma drug that will be administered in single doses (Part 1) and repeated doses (Parts 2 and 3), using either a nebulizer or dry powder inhaler (DPI). As part of the investigation, a single cohort of healthy volunteers who previously took inhaled study medication will also be subject to intravenous (IV) administration of study medication (Part 1b).

    The study drug is being developed by AstraZeneca, for treatment of patients with moderate to severe asthma. Researchers foresee that the study drug will decrease overall inflammation and reduce episodes of worsening of symptoms, with accompanying improvement of lung function.

    Each study part will include a screening visit, a treatment period and a follow-up visit. Eligible participants will remain residential at the Clinical Unit for the full duration of the treatment period.

    This is a first-in-human clinical trial. Conditional inclusion of women of non-childbearing potential is allowed in this study. The main purpose of the study is to see how safe the study drug is and how well the body tolerates the study drug after single and repeated doses, administered by inhalation. The study will also investigate how the study drug is absorbed (taken up into the body), metabolised (chemically broken down), distributed through the body, and excreted (removed from the body) (overall referred to as PK). In addition, the study will investigate the anti-inflammatory effect as a measure of the effects of the study drug on the body (referred to as pharmacodynamics [PD]) and the way in which the study drug works (mechanism of action).

    Summary of Results
    The lay summary of study results is under preparation and will be posted on https://eur03.safelinks.protection.outlook.com/?url=http%3A%2F%2Fwww.trialsummaries.com%2F&data=05%7C01%7Capprovals%40hra.nhs.uk%7C26977fb0dd784dcbe09008da8f6aa522%7C8e1f0acad87d4f20939e36243d574267%7C0%7C0%7C637979985463671250%7CUnknown%7CTWFpbGZsb3d8eyJWIjoiMC4wLjAwMDAiLCJQIjoiV2luMzIiLCJBTiI6Ik1haWwiLCJXVCI6Mn0%3D%7C3000%7C%7C%7C&sdata=h0%2FgklzwqrC4cd%2BqU6cSPOgdJKYruBu8DxulSsto2Bc%3D&reserved=0 within 2 years of study end.

  • REC name

    London - London Bridge Research Ethics Committee

  • REC reference

    18/LO/1432

  • Date of REC Opinion

    14 Nov 2018

  • REC opinion

    Further Information Favourable Opinion