A study to assess the mass balance of TAK-385 in HVs (QBR117173)

  • Research type

    Research Study

  • Full title

    An Open Label, Single Centre, Two Part Phase I Mass Balance Study to Assess the Absorption, Distribution, Metabolism, Excretion and Absolute Bioavailability of Orally Administered [14C]-TAK-385 in Healthy Male Subjects

  • IRAS ID

    159818

  • Contact name

    Pui Leung

  • Contact email

    pui.leung@quotientclinical.com

  • Sponsor organisation

    Takeda Development Centre Europe Ltd.

  • Eudract number

    2014-001564-35

  • Research summary

    TAK-385 is being developed by the sponsor and is undergoing parallel clinical development as a potential treatment for gynaecological conditions in women, such as heavy menstrual bleeding and fibroids, and prostate cancer in men.

    The purpose of this 2 part study is to look at how TAK-385 is taken up, broken down and removed from the body when given as a radiolabelled oral solution (by mouth), or as an oral tablet (by mouth) followed by a radiolabelled intravenous infusion into the arm vein.

    The study will consist of 2 parts involving up to 12 healthy male subjects. In Part 1, up to 6 subjects will receive a single 80 mg dose of [14C]-TAK-385 administered as an oral solution. In Part 2, up to 6 subjects will receive a single oral 80mg dose of TAK-385 administered as two 40mg tablets and an 80µg intravenous (into a vein) dose of [14C]-TAK-385

  • REC name

    Wales REC 2

  • REC reference

    14/WA/1087

  • Date of REC Opinion

    3 Sep 2014

  • REC opinion

    Further Information Favourable Opinion