A Phase I study of Y14 in adult subjects

  • Research type

    Research Study

  • Full title

    A randomised, placebo controlled first in human study to investigate the safety, tolerability, pharmacokinetics and pharmacodynamics of Y14 in adult subjects

  • IRAS ID

    222848

  • Contact name

    Jim Bush

  • Contact email

    Jim.Bush@covance.com

  • Sponsor organisation

    Imperial College London| Imperial College Healthcare NHS Trust

  • Eudract number

    2017-000380-33

  • Clinicaltrials.gov Identifier

    NCT03673111

  • Clinicaltrials.gov Identifier

    REC, 17/NW/0084

  • Duration of Study in the UK

    1 years, 0 months, 3 days

  • Research summary

    Y14 is a new molecule, being developed as a treatment for obesity. Y14 binds to the Y2 receptor causing increased satiety (feelings of fullness after eating) and reduced body weight. There are licenced drugs with similar mechanisms of action, it is hoped that Y14 will have a greater duration of action and a better side-effect profile.

    The main purpose of this first in man study is to assess safety and tolerability when Y14 is given as a SC (Subcutaneous, under the skin) injection. Other objectives include an assessment of the pharmacokinetics of the drug (how quickly the drug gets into the blood stream and how quickly it is removed from the body). An assessment of effects on food consumption, body weight hormone levels and glucose levels.

    This study will be conducted in two parts. Part A will be a single dose study, in 5 cohorts of overweight but otherwise healthy subjects. Cohort 1 will consist of 4 subjects (3 active drug, 1 placebo (dummy drug). Each subject in cohort 1 will receive 3 single doses of drug at different dose levels. Cohort 2 onwards will consist of 6 subjects (5 active, 1 placebo) and each subject will be dosed once only. The first two subjects in cohort 1 will be dosed 1 week before the rest of the cohort on the first dosing occasion. For the second and third doses all subjects will be dosed on the same day. Part B will be a multiple dose study in patients with diabetes or pre-diabetes. Three dose levels will be tested in 3 cohorts, each of 8 subjects (6 active, 2 placebo Subjects will receive 5 doses of Y14 or placebo each separated by 7 days. Additional cohorts may be enrolled; up to 8 in Part A and 3 in Part B.

  • REC name

    North West - Greater Manchester Central Research Ethics Committee

  • REC reference

    17/NW/0084

  • Date of REC Opinion

    22 Mar 2017

  • REC opinion

    Favourable Opinion